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九州大学大学院薬学研究院
環境調和創薬化学分野
Green Pharmaceutical Chemistry
Graduate School of Pharmaceutical Sciences, Kyushu University

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2017

Zhao Li, Masamichi Tamura, Ryo Yazaki, Takashi Ohshima
Catalytic Chemoselective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Ester: Hydroxy Group over Amino Group and Conjugate Addition over Transesterification
Chem. Pharm. Bull. 2017, 65, 19–21. DOI: 10.1248/cpb.c16-00333
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Kazuhiro Morisaki, Hiroyuki Morimoto, Kazushi Mashima, and Takashi Ohshima
Direct Enantioselective Alkynylation of α-Ketoesters and α-Ketiminoesters Catalyzed by [Bis(oxazoline)phenyl]rhodium(III) Complexes
Heterocycles 2017, 95, 637661. DOI:10.3987/REV-16-SR(S)4
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Ren-Shi Li, Tomoki Takeda, Takashi Ohshima, Hideyuki Yamada, Yuji Ishii
Metabolomic profiling of brain tissues of mice chronically exposed to heroin
Drug Metabolism and Pharmacokinetics 2017, 32, 108–111. DOI: 10.1016/j.dmpk.2016.10.410

Toru Deguchi, Hai-Long Xin, Hiroyuki Morimoto, and Takashi Ohshima
Direct Catalytic Alcoholysis of Unactivated 8-Aminoquinoline Amides
ACS Catal. 2017, 7, 3157–3161. DOI: 10.1021/acscatal.7b00442
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Kazuhiro Morisaki, Hiroyuki Morimoto and Takashi Ohshima
Direct access to N-unprotected tetrasubstituted propargylamines via direct catalytic alkynylation of N-unprotected trifluoromethyl ketimines
Chem. Commun. 2017, 53, 6319–6322. DOI: 10.1039/C7CC02194A (Press Release, Highlighted by Chem-Station) (Backcover)
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Seiya Taninokuchi, Ryo Yazaki and Takashi Ohshima
Catalytic Aerobic Chemoselective α-Oxidation of Acylpyrazoles en Route to α-Hydroxy Acid Derivatives
Org. Lett. 2017, 19, 3187–3190. DOI: 10.1021/acs.orglett.7b01293
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Masanao Sawa, Kazuhiro Morisaki, Yuta Kondo, Hiroyuki Morimoto and Takashi Ohshima
Direct Access to N-Unprotected α- and/or β-Tetrasubstituted Amino Acid Esters via Direct Catalytic Mannich-Type Reactions Using N-Unprotected Trifluoromethyl Ketimines
Chem. Eur. J. 2017 Early View. DOI: 10.1002/chem.201703516 (Press Release) (Cover Picture, DOI: 10.1002/chem.201704439)
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Amrita Das, Kenji Watanabe, Hiroyuki Morimoto and Takashi Ohshima
Boronic Acid Accelerated Three-Component Reaction for the Synthesis of α-Sulfanyl-Substituted Indole-3-acetic Acids
Org. Lett. 2017, Article ASAP. DOI: 10.1021/acs.orglett.7b02727
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Kazuhiro Morisaki, Yuta Kondo, Masanao Sawa, Hiroyuki Morimoto, Takashi Ohshima
Synthesis of 1-Tetrasubstituted 2,2,2-Trifluoroethylamine Derivatives via Palladium-Catalyzed Allylation of sp3 C–H Bonds
Chem. Pharm. Bull. 2017, 65, 1089–1092. DOI: 10.1248/cpb.c17-00580
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